Mofuta o moholo oa Tianeptine hemisulfate monohydrate powder (1224690-84-9)

October 30, 2018

Tianeptine Sulfate, eo hape e bitsoang Raw Tianeptine hemisulfate monohydrate powder, ke …… ..


Boemo: Ka Phatlalatso ea Mesebetsi
Sehlopha: 25kg / Drum
Bokhoni: 1350kg / khoeli

Pure ea heaneptine ea hemisptate monohydrate powder (1224690-84-9) video

 

Mahlaseli a mangata a heaneptine a hemisulfate monohydrate (1224690-84-9) Lintlha

Name Product Mofuta o moholo oa Tianeptine hemisulfate monohydrate powder
Lebitso la lik'hemik'hale Tianeptine hemisulfate monohydrate; 1224690-84-9; Heptanoic acid,
Brand Name Stablon, Coaxil
Sehlopha sa Lithethefatsi Lipakeng le Lik'hemik'hale tse Ntle
Nomoro ea CAS 1224690-84-9
InChIKey KVVMXNNJBVTOSX-UHFFFAOYSA-N
limolek'hule Formula C42H56Cl2N4O14S3
limolek'hule Wtse robeli 1008.004 g / mol
Masapo a monoisotopic 1006.233 g / mol
Ho qhibiliha Poli  1800 ° C
Ho belisoa Poli 269.8 ° C ho 760 mmHg
Likokoana-hloko tsa Half-Life N / A
Color Phofshoana e ntle
Sho khoneha  Ho qhibiliha ka metsi ka metsing le methanol le dichloromethane
Storage Tmocheso  Sebaka se omileng se pholileng
Aho latela Sesedium ea Tianeptine e ka sebelisoa Tricyclic e nang le psychostimulant

Sodium ea Tianeptine e na le mesebetsi ea ho loantša seso le anti-emetic. Ho tepella maikutlo

 

Mofuta o moholo oa Tianeptine hemisulfate monohydrate (THM) powder (1224690-84-9)

Mofuta o moholo oa Tianeptine hemisulfate monohydrate powder, eo hape e bitsoangTianeptine Sulfate, ke phetoho e ntlafetseng ea foromo ea letsoai ea sodium ea soane. Ha e hloekile, e bonolo ho sebetsana le eona, e theoha fatše, ebile e nka habeli ka nako e telele. E na le melemo e tšoanang le e kang Sodium ea Tianeptine, mofuta oa sulfate feela o na le halofo ea lihora tsa 5-6, kahoo e nka habeli ka nako e telele joaloka sodium ea tianeptine. Ka lebaka la sena, bafuputsi ba tla hloka linako tsa 2-3 palo ea sulfate ho finyella liphello tseo ba li ratang ho tloha sodium. Sulfate e boetse e fokotseha haholo ka bobeli le litlolo.

Heaneptine hemisulfate monohydrate e khethoa e le serotonin reuptake enhancer (SSRE) e sebelisoang ho tšoara khatello ea maikutlo. Tianeptine e ile ea hlahisoa Fora ho 1960s 'me e sebelisitsoe hohle karolo ea ho qetela ea 2000s.

Hape ka linako tse ling ho sebelisoa ho tšoara lefu la sefuba kapa lefu la masapo. Ha ho etsoa litekanyetso tse boima ho tlalehoa hore ho hlahisa liphello tse kang tsa sediti le ho tsosolosa, ho ntlafatsa tšusumetso le ho thaba ha li laoloa.

Tianeptine hemisptate monohydrate (THM) powder (1224690-84-9) Mehato ea Liketso

E 'ngoe ea mekhoa ea mantlha ea ts'ebetso ea Tianeptine hemisulfate monohydrate ke ho eketsa ts'ebetso ea serotonin (5-HT) bokong le liplatelete. Ho fapana le metsoako e mengata ea tricyclic, Tianeptine ha e bonahale e amahanngoa le ho fokotseha ha ts'ebetso ea ts'ebetso kapa ts'ebetso ea makoloi. Ho bonahala e na le ts'ebetso ho sistimi ea glutamatergic, eo ho nahanoang hore ke mokhoa oa ho loants'a khatello ea maikutlo.

Ka ho eketsa ts'ebeliso ea serotonin, Tianeptine hemisulfate monohydrate e na le mochini o fapaneng le oa li-SSRI tsa setso. Liphuputso tsa morao-rao li hlahlobile litlamorao tsa Tianeptine kahare ho mohopolo oa neuroplasticity oa khatello ea maikutlo, moo e ka bang le ts'ebetso e itseng. Liphuputso tsa morao-rao li bonts'a hore Tianeptine e kanna ea sebelisana le adenosine A1 receptors.

Ho feta moo, lipatlisiso tsa morao-rao tse phatlalalitsoeng ho 2014 li bontša hore Tianeptine e ka sebetsa joaloka m-opioid receptor (MOR) agonist. Bafuputsi ba ile ba sebelisa li-radioligand tse tlamang le li-cell-based test assays ho tseba Tianeptine e le MOR agonist e sebetsang hantle. Hape ke agonist e feletseng ea opioid empa ka kamano e tlaase haholo. Tianeptine e ne e sa sebetse libakeng tsa k-opioid receptor.

tshebediso ea Tianeptine hemisptate monohydrate (THM) powder (1224690-84-9)

▪ Ho tepella maikutlo

▪ Litšoaneleho tsa khatello ea maikutlo le khatello ea maikutlo le nootropic

▪ Mosebetsi oa kutloisiso le bokhoni bo ntlafetseng ba ho ithuta

▪ Bohloko ba mesifa

▪ ADHD

Ho khothalletsoa Tianeptine hemisptate monohydrate (THM) powder (1224690-84-9) Palo

Tekanyo ea tianeptine hemisulfate monohydrate hangata e 25 mg hang, kapa habeli ka letsatsi. Le ha o qala ka litekanyetso tse tlase, ho molemo ho e fokotsa ho matsatsi a 2 kapa a 3 ka beke bonyane matsatsi a 3 - 4 mahareng.

Tianeptine hemisulfate monohydrate e tla ka sebopeho sa capsule kapa phofo. Ho kgothaletswa ho qala ka litekanyetso tse tlase ebe o eketseha ka nyane ho fihlela tekanyetso e nepahetseng e fumaneha. Ntle le moo, litekanyetso tse nyane li fokotsa monyetla oa ho lemalla, ho tlohela haholo, le mamello.

Tekanyo ea 50-75 mg e ka ba e hlasimollang. Tekanyo ea boithabiso ea Tianeptine hemisulfate monohydrate ea> 100 mg e ka baka maikutlo a phahameng a Tianeptine hemisulfate monohydrate.

Melemo ea Tianeptine hemisptate monohydrate (THM) powder (1224690-84-9)

♦ Tianeptine hemisulfate monohydrate e ntlafatsa bokong ba pelo le ho fokotsa khatello ea maikutlo. Neuroplasticity ke bokhoni ba boko ba ho ikamahanya le ho fetoha ha o ithuta; ho kenya letsoho mosebetsing o ntlafetseng oa tsebo le bokhoni bo ntlafetseng ba ho ithuta.

Phuputso ea bakuli ba 90 ba nang le PTSD e bontšitse litholoana tse ntle ka ts'ebeliso ea Tianeptine hemisulfate monohydrate. Boithuto bo boetse bo bontšitse hore ka kalafo ea tianeptine sulfate le phokotso e kholo ea ts'abo ea ts'abo. Tianeptine hemisulfate monohydrate e fuoeng bakuli ba seng ba tsofetse e bonts'itse ho ntlafatsa ts'ebetso ea khatello ea kelello le ntlafatso ea maikutlo.

• Lithuto tsa liphoofolo le tsa batho li 'nile tsa etsoa kalafo ea Parkinson le lefu la Tianeptine hemisulfate monohydrate, e bontšang liphello tse tšepisang ho ntlafatsa lintlha tsa bophelo bo botle ba kelello.

Phuputso ea pele ea bakuli ba 68 ba nang le ADHD e fihletse qeto ea hore lipalo tse bolelang li ntlafalitse haholo le hore Tianeptine hemisulfate monohydrate e na le molemo ho nolofalletsa bokhoni ba ho ela hloko le ho fokotsa boits'oaro bo sa sebetseng.

♦ Tianeptine hemisulfate monohydrate hape ke analgesic e sebetsang hantle (painkiller), esita le bakeng sa batho ba nang le bohloko bo sa foleng. Ke mokhoa o atlehang oa ho fokotsa matšoao a amanang le mathata a bophelo ba mala.

♦ Setsi sa Teko ea Bongaka sa Caracas se ile sa etsa liteko tsa bana ba nang le asthma libeke tse 52. Bakuli ba fuoeng Tianeptine hemisulfate monohydrate ba bontšitse keketseho e kholo ts'ebetsong ea matšoafo.

• Le hoja ho hlokahala lipatlisiso tse ngata, ho ithuta ha banna ba 237 le ED ho entse qeto ea hore tianeptine e ka ba phekolo e sebetsang.

• Matšoao a Tianeptine a khatello ea kelello ha a na tšusumetso e mpe ea acetylcholine kapa lefu la pelo, ho etsa tianeptine khetho e babatsehang bakeng sa ba tsofetseng hammoho le tse ling