Raw YK-11 phofo (431579-34-9) video
Raw YK-11 phofo (431579-34-9) Tlhaloso
YK11, e tsejoang hape e le Myostine, e nkoa e le e 'ngoe ea phofo e matla ea YK11' marakeng. Ke moetsi oa li-androgen receptor ea maiketsetso ea maiketsetso. Setlhare se na le ts'ebetso ea anabolic ho vitro ho C2C12 myoblasts mme e bonts'a potency e kholo ho feta dihydrotestosterone (DHT) ntlheng ena. YK11 hape ke inhibitor ea Myostatin. ba ka u thusa ho fumana mesifa le ho lahleheloa ke mafura.
Raw YK-11 phofo (431579-34-9) Slitšobotsi
Name Product | Raw YK-11 phofo |
Lebitso la lik'hemik'hale | YK11, (17a, 20E) -17,20 - [(1-Methoxyethylidene) bis (oxy)] - 3-oxo-19-norpregna- 4,20-diene-21-carboxylic Acid Methyl Ester; YK11 ((17A, 20E) -17,20 - [(1-methoxyethylidene) bis- (oxy)] - 3-oxo-; DNA (Terrabacter strain YK11 16S rRNA gene fragment); GenBank AB070463 |
Brand Name | Ha ho data e fumanehang |
Sehlopha sa Lithethefatsi | YK11 phofo |
Nomoro ea CAS | 431579-34-9 |
InChIKey | KCQHQCDHFVGNMK-DEIKBOPOSA-N |
limolek'hule Formula | C25H34O6 |
limolek'hule Wtse robeli | 430.53386 |
Masapo a monoisotopic | 430.236 g / mol |
Ho qhibiliha Poli | 190-200 ° C |
Fho tsosolosa Poli | Ha ho data e fumanehang |
Likokoana-hloko tsa Half-Life | Lihora tsa 6-10, ho itšetlehile ka motho ka mong |
Color | Tšepe e tšoeu |
Sho khoneha | Propylene Glycol, DMSO, Ethanol |
Storage Tmocheso | Mocheso oa kamore |
Raw YK-11 phofo Aho latela | Selection Androgen Receptor Modulator, Myostatin Inhibitor |
Raw Raw YK-11 phofo (431579-34-9) Tlhaloso
Basebelisi ba bangata ba nahana hore YK11 ke senotlolo sa ho notlolla bokhoni ba 'mele ka botlalo le ho fumana melemo ea mesifa e potlakileng ka litla-morao tse fokolang. E boetse ea re YK11 e na le bokhoni ba ho fokotsa ts'ebetso ea myostatin, e e etsa myostatin inhibitor. YK-11 ehlile ke e 'ngoe ea tse matla ho fetisisa ka ntle mono. U ke ke ua bapisa YK le LGD-4033 kapa lihlahisoa tse ling ka lebaka la matla a eona.
Leha ho le joalo, leha phofo e tala ea YK-11 e le matla ka mokhoa o makatsang hopola hore ho bile le lithuto tse 'maloa tse entsoeng ka komporo ena. Lena ke lona lebaka le ka sehloohong batho ba bangata ba bonahalang ba khetha ho ea le ba bang ba kang Ostamuscle, RAD-140 kapa GW-501516.
YK11 e fumana phaello ho lihahi tsa 'mele ka lebaka la bokhoni ba eona ba ho haha mesifa kapele le litlamorao tse fokolang.
Thuto e 'ngoe ea lisele e bontša hore YK11 e eketsa mesifa ea mesifa. Bafuputsi ba fumane hore ho eketsa protheine ea follyatin follistatin (a myostatin inhibitor).
YK11 e ka boela ea eketsa bophelo bo botle ba masapo. Phuputsong ea masapo a masapo, YK11 e ile ea eketsa litekanyetso tsa liprotheine tsa ho haha masapo.
Ba bang ba 'mele ba ileng ba leka YK11 ba tlaleha melemo e mengata ea mesifa le tahlehelo ea mafura le liphello tse fokolang. Leha ho le joalo, hona joale ha ho na liphoofolo kapa lithuto tsa batho tsa YK11 le tšireletseho ea eona e sa hlaka.
Raw YK-11 phofo (431579-34-9) Mokhoa oa Ketso
YK11 e na le lik'hemik'hale tse tšoanang le tsa DHT 'me sena se bontšoa ka tsela eo e tlamang li-receptor tsa androgen. 'Mele o hlahisa DHT ka tlhaho ka morero oa ho khothalletsa bophelo bo botle ba prostate, kholo ea moriri, le tsoelo-pele e loketseng ea bokhachane.
Bafuputsi ba ile ba etsa phuputso ea sele ho fumana hore na e sebetsa joang ho haha mesifa. Liphetho li bontša hore e ikemiselitse ho eketsa maemo a follistatin. Follistatin ke e 'ngoe ea protheine e tloaelehileng' meleng oa motho e thusang ho boloka myostatin ho hlahloba. Myostatin ke hormone eo mosebetsi oa eona e leng ho fokotsa mesifa e sa tsitsang.
Ho fihlela joale, feela YK11 phofo e tala e na le matla a ho thibela myostatin.
Bopaki bo bong bo fana ka maikutlo a hore YK11 e ka boela ea khothalletsa kholo ea bone ka ho kena-kenana le monyako o sebetsang joaloka DHT.
melemo e ea Raw YK11 phofo (431579-34-9)
E eketsa boholo ba mesifa
YK11 e na le bokhoni bo makatsang ba ho tsosa kholo ea mesifa.
Ke hobane ka tlhaho ho eketsa menyetla ea follistatin eo hape e ntlafatsang bokhoni ba 'mele oa hao oa ho hlahisa lisele tsa mesifa. Follistatin e boetse e na le boikarabello ba ho thibela myostatin, ka tsela eo ho u bula ho fihlela monyetla oa ho ba le mesifa e sa felleng. Empa haeba liphello tsa follistatin li thibeloa ka tsela leha e le efe, joale ho thibela myostatin ho ke ke ha etsahala, e leng ho ka etsang hore YK11 e se ke ea atleha.
Hase ho utloahala joaloka tlaleho e robehileng empa ha ho na lithuto tsa batho kapa tsa liphoofolo ho khutlisetsa boitsebiso boemong bona.
Sohle seo re nang le sona ke bopaki ba anecdotal bo thehiloeng ho liphuputso tsa 'mele ka liforomo tsa inthanete. Seo ba re bolellang sona ke hore ba khonne ho fokotseha haholo mafura le li-lbs tsa 15 tsa bohlokoa tsa mesifa e boima ka nako e khutšoanyane.
E Matlafatsa Masapo
Lihormone tsa thobalano li bohlokoa bakeng sa ho boloka masapo a matla le a phetseng hantle. Bopaki bo fumanehang bo bontša hore YK11 phofo e tala e ka eketsa matla a masapo ka ho itlama ho li-androgen receptors.
YK11 e ka boela ea eketsa boholo ba PKB (protein kinase B) e fumanehang lisele tsa 'mele tse thusang ho hōla ha lisele tsa masapo.
A re se keng ra lebala hore o batla ho ba le mesifa le masapo a matla, a phetseng hantle ho qoba fractures. E ka 'na ea khona ho thusa tabeng ena hape hobane e atleha haholo ho haha mesifa, ho tšehetsa bophelo bo botle ba masapo le ho fokotsa liphello tsa lesapo la masapo.
Motsoako o motsoako oa YK-11 (431579-34-9).
Baetsi ba 'mele ba sebelisitseng phofo e tala ea YK11 ba re ho e nka ka litekanyetso tsa 10 ho isa ho 15 mg ka letsatsi ho ba sebeletsa hantle. Ba bang ba tlalehile litlamorao tse ntle ho 5 mg ka letsatsi. Basebelisi ba bangata ba e potoloha libeke tse 4 ho isa ho tse 8.
Litla-morao tsa Raw YK-11 phofo (431579-34-9)
▲ Hona joale, lithuto tsa lisele feela li 'nile tsa khannoa ka YK11.
Ha ho na bopaki ba bongaka kapa esita le lithuto tsa liphoofolo ho khutlisa lipolelo tse ling tse ntseng li etsoa ka moriana.
Sena se lokela ho etsa hore o nahane ka makhetlo a mabeli ka lipatlisiso ka likarolo tsena. Mohlomong u lokela ho hlahloba lik'hemik'hale tse sa tšoaneng tse kang Ostarine le Ligandrol. Ba na le boitsebiso bo bongata le lipatlisiso tse teng.
Ho boleloa hore YK11 e ka ba chefo ho sebete. Ha e bua ka mokhoa oa ho itlhakisa, e ka ama kholo ea moriri, khoele ea mantsoe, bophelo ba senya le likarolo tse ling tsa bohlokoa 'meleng.